Synthesis of tritium-labeled levetiracetam ((2S)-2-(2-oxopyrrolidin-1-yl) butanamide) with high specific activity

Simone Hildenbrand; Younis Baqi; Christa E. Müller

doi:10.1002/jlcr.1942

Synthesis of tritium-labeled levetiracetam ((2S)-2-(2-oxopyrrolidin-1-yl) butanamide) with high specific activity

Simone Hildenbrand, Younis Baqi, Christa E. Müller^*

^*المؤلف المقابل لهذا العمل

نتاج البحث: المساهمة في مجلة › Article › مراجعة النظراء

4 اقتباسات (Scopus)

ملخص

A method for the preparation of [Â³H]levetiracetam with a high specific activity of 98Ci/mmol (3.6TBq/mmol) is described. The radioligand proved to be highly useful for the labeling of specific levetiracetam binding sites in rat brain membrane preparations.

اللغة الأصلية	English
الصفحات (من إلى)	48-51
عدد الصفحات	4
دورية	Journal of Labelled Compounds and Radiopharmaceuticals
مستوى الصوت	55
رقم الإصدار	1
المعرِّفات الرقمية للأشياء	https://doi.org/10.1002/jlcr.1942
حالة النشر	Published - يناير 2012
منشور خارجيًا	نعم

ASJC Scopus subject areas

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الوصول إلى المستند

10.1002/jlcr.1942

الملفات والروابط الأخرى

قم بذكر هذا

Synthesis of tritium-labeled levetiracetam ((2S)-2-(2-oxopyrrolidin-1-yl) butanamide) with high specific activity. / Hildenbrand, Simone; Baqi, Younis; Müller, Christa E.
في: Journal of Labelled Compounds and Radiopharmaceuticals, المجلد 55, رقم 1, ٠١.٢٠١٢, صفحة 48-51.

نتاج البحث: المساهمة في مجلة › Article › مراجعة النظراء

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abstract = "A method for the preparation of [{\^A}3H]levetiracetam with a high specific activity of 98Ci/mmol (3.6TBq/mmol) is described. The radioligand proved to be highly useful for the labeling of specific levetiracetam binding sites in rat brain membrane preparations.",

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Synthesis of tritium-labeled levetiracetam ((2S)-2-(2-oxopyrrolidin-1-yl) butanamide) with high specific activity

ملخص

ASJC Scopus subject areas

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